PF-04628935
Product Specifications
CAS Number
1383719-97-8
Target
GHSR|||Others
Related Pathways
GPCR/G Protein|||Others
Bioactivity
PF-04628935 is a potent antagonist/inverse agonist of the ghrelin receptor, growth hormone secretagogue receptor 1a (GHS-R1a) with an IC50 of 4.6 nM. PF-04628935 is orally bioavailable and brain penetrant.
Smiles
C(N1CC2(C1)CCN(C(CC3=CN4C(=N3)SC(C)=C4)=O)CC2)C5=C(Cl)C=C(C=C5)N6N=CC=N6
Molecular Formula
C24H26ClN7OS
Molecular Weight
496.03
Shipping Conditions
Cool pack
Storage Temperature
-20°C
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