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PD 174265

Product Specifications

CAS Number

216163-53-0

Target

EGFR

Related Pathways

Angiogenesis|||JAK/STAT signaling|||Tyrosine Kinase/Adaptors

Purity

0.9951

Bioactivity

PD 174265 is an effective, selective and reversible inhibitor of epidermal growth factor receptor (EGFR) with an IC50 of 0.45 nM.

Smiles

CCC(=O)Nc1ccc2ncnc(Nc3cccc(Br)c3)c2c1

Molecular Formula

C17H15BrN4O

Molecular Weight

371.23

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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