NNC052090
Product Specifications
CAS Number
184845-43-0
Target
Others, GABA Receptor
Related Pathways
Membrane transporter/Ion channel, Others, Neuroscience
Bioactivity
NNC052090 is a GABA uptake inhibitor that displays moderate selectivity for BGT-1 transporters with Ki values are 1.4, 15, 19 and 41 μM for hBGT-1, hGAT-3, hGAT-1 and hGAT-2 respectively. NNC052090 also displays affinity at α1- and D2-receptors with IC50 values are 266 and 1632 nM respectively.
Smiles
C(CCN1CCC(O)(CC1)C2=C(OC)C=CC=C2)N3C=4C(C=5C3=CC=CC5)=CC=CC4
Molecular Formula
C27H30N2O2
Molecular Weight
414.54
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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