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MPX-007

Product Specifications

CAS Number

1688685-29-1

Target

Others|||iGluR

Related Pathways

Others|||Neuroscience|||Membrane transporter/Ion channel

Bioactivity

MPX-007, a potent NMDA inhibitor, inhibits GluN2A-containing NMDA receptors expressed in HEK cells with IC50s of 27 nM.

Smiles

C(NS(=O)(=O)C1=CC(F)=C(F)C=C1)C=2C(C)=NC(C(NCC=3SC(C)=NC3)=O)=CN2

Molecular Formula

C18H17F2N5O3S2

Molecular Weight

453.49

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

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