FT001
Product Specifications
CAS Number
1778655-51-8
Target
Epigenetic Reader Domain
Related Pathways
Chromatin/Epigenetic
Purity
>99.99%
Bioactivity
FT001 is a potent, selective and orally available inhibitor of BET Bromodomain with antitumor activity. FT001 inhibited the expression of MYC with the IC50 value of 0.46 μM) . FT001 has potent antiproliferative effects against MV-4-11 and demonstrates significant MYC mRNA suppression both in vitro and in vivo.
Smiles
C(=O)(N1C=2C(N(C(C)=O)[C@@H](C)C1)=CC=C(C2)C3=CC=C(C=C3)N4CCS(=O)(=O)CC4)C5CC5
Molecular Formula
C25H29N3O4S
Molecular Weight
467.58
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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