CP 154,526

157286-86-7

Others|||CRFR

GPCR/G Protein|||Others

CP 154,526 is a selective CRF1 receptor antagonist (Ki = 2.7 nM) . CP 154,526 blocks CRF-induced activation of adenylate cyclase and the HPA axis.

N(CCCC)(CC)C1=C2C(N(C=C2C)C3=C(C)C=C(C)C=C3C)=NC(C)=N1

C23H32N4

364.53

Cool pack

-20°C