CJ-15208
Product Specifications
CAS Number
210236-47-8
Target
Others, Opioid Receptor
Related Pathways
Endocrinology/Hormones, Neuroscience, GPCR/G Protein, Others
Bioactivity
CJ-15208 is a potent and selective κ-opioid receptor antagonist from a fungus, Ctenomyces serratus ATCC15502 (IC50 are 47 nM for kappa, 260 nM for mu, and 2,600 nM for delta respectly) . In the electrically-stimulated twitch response assay of rabbit vas deferens, CJ-15208 recovered the suppression by a kappa agonist asimadoline with an ED50 of 1.3 microM.
Smiles
C(C=1C=2C(NC1)=CC=CC2)[C@H]3C(=O)N[C@@H](CC4=CC=CC=C4)C(=O)N5[C@@](C(=O)N[C@@H](CC6=CC=CC=C6)C(=O)N3)(CCC5)[H]
Molecular Formula
C34H35N5O4
Molecular Weight
577.67
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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