BMS-986122
Product Specifications
CAS Number
313669-88-4
Target
Opioid Receptor
Related Pathways
Neuroscience, Endocrinology/Hormones, GPCR/G Protein
Purity
0.9986
Bioactivity
BMS-986122 (BMS 986122) is a positive allosteric modulator of μ-opioid receptors that increases β-arrestin recruitment stimulated by endomorphin 1 in U2OS-OPRM1 human osteosarcoma cells expressing μ-opioid receptors (EC50 = 3 μM) .
Smiles
COc1ccc(cc1Br)C1SCCN1S(=O)(=O)c1ccc(Cl)cc1
Molecular Formula
C16H15BrClNO3S2
Molecular Weight
448.78
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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