GSK2656157
Product Specifications
CAS Number
1337532-29-2
Target
Autophagy, Apoptosis, PERK
Related Pathways
Autophagy, Apoptosis
Purity
>99.99%
Bioactivity
GSK2656157 is a highly specific and ATP-competitive PERK inhibitor (IC50: 0.9 nM) in a cell-free assay. The selectivty is 500-fold higher against a panel of 300 kinases.
Smiles
Cc1cccc(CC(=O)N2CCc3c2ccc(-c2cn(C)c4ncnc(N)c24)c3F)n1
Molecular Formula
C23H21FN6O
Molecular Weight
416.45
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog