What is the catalog number for Ici 216140?

The catalog number for Ici 216140 is T25522.

What sizes are available for Ici 216140?

Ici 216140 is available in the following size(s): 500 µg, 1 mg, 5 mg.

How many pack sizes does Ici 216140 come in?

Ici 216140 is available in 3 different pack sizes.

Is Ici 216140 in stock?

Ici 216140 is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures Ici 216140?

Ici 216140 is manufactured by Molfinity.

What is the estimated delivery time for Ici 216140?

Estimated delivery time for Ici 216140 is approximately 10 business day(s), depending on your location.

Ici 216140

Product Specifications

CAS Number

124001-41-8

Target

Others, Bombesin Receptor

Related Pathways

Others, GPCR/G Protein

Bioactivity

ICI 216140 is a GRP/bombesin receptor 2 antagonist (IC50: 2 nM in vitro) . At 2 mg/kg, it can decrease bombesin-stimulated pancreatic amylase secretion in rats. At 1 mM, it has been proved to attenuate bombesin-stimulated increases in blood pressure in rats.

Smiles

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