Dersimelagon
Product Specifications
CAS Number
1835256-48-8
Target
Melanocortin Receptor
Related Pathways
Neuroscience, GPCR/G Protein
Purity
0.9823
Bioactivity
Dersimelagon (MT-7117) is an orally active, selective melanocortin 1 receptor (MC1R) agonist with EC50 values of 8.16, 3.91, 1.14, and 0.251 nM for human (h), cynomolgus monkey (cm), mouse (m), and rat (r) MC1R, respectively. Dersimelagon exhibits good affinity for hMC1R and hMC4R, with Ki values of 2.26 and 32.9 nM, respectively. Dersimelagon can be used in the study of skin pigmentation[1].
Smiles
C(=O)([C@@]1(F)[C@@H](CN(C1)C2CCCC2)C3=CC=C(OC)C=C3)N4C[C@@H]([C@@H](COC)C4)C5=C(C=C(C(F)(F)F)C=C5)N6CCC(C(O)=O)CC6
Molecular Formula
C36H45F4N3O5
Molecular Weight
675.75
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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