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Galunisertib

Product Specifications

CAS Number

700874-72-2

Target

TGF-beta/Smad

Related Pathways

Stem Cells

Purity

>99.99%

Bioactivity

Galunisertib (LY2157299) is a TGF-β receptor type I (TGF-βRI) inhibitor (IC50=56 nM) that is selective. Galunisertib has antitumor activity and can be used in combination with PD-1 inhibitors.

Smiles

Cc1cccc(n1)-c1nn2CCCc2c1-c1ccnc2ccc(cc12)C(N)=O

Molecular Formula

C22H19N5O

Molecular Weight

369.42

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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