Galunisertib
Product Specifications
CAS Number
700874-72-2
Target
TGF-beta/Smad
Related Pathways
Stem Cells
Purity
>99.99%
Bioactivity
Galunisertib (LY2157299) is a TGF-β receptor type I (TGF-βRI) inhibitor (IC50=56 nM) that is selective. Galunisertib has antitumor activity and can be used in combination with PD-1 inhibitors.
Smiles
Cc1cccc(n1)-c1nn2CCCc2c1-c1ccnc2ccc(cc12)C(N)=O
Molecular Formula
C22H19N5O
Molecular Weight
369.42
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog