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PF-06807656

Product Specifications

Target

Others

Related Pathways

Others

Bioactivity

PF-06807656 is insensitive to the introduction of the N171D mutation in the ROMK conduction pore that greatly diminishes the activity of other small-molecule inhibitors. PF-06807656 is an effective ROMK inhibitor (Tl+ flux IC50 = 160 nM) .

Smiles

O=C(NC(C1=NN(C)N=C1)C)C2=CC(S(=O)(NC3=CC=C(Cl)C=C3)=O)=C(OC)C=C2

Molecular Formula

C19H20ClN5O4S

Molecular Weight

449.91

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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