EPZ011989
Product Specifications
CAS Number
1598383-40-4
Target
Histone Methyltransferase
Related Pathways
Chromatin/Epigenetic
Purity
0.9981
Bioactivity
EPZ011989 is a effective, specific orally bioavailable EZH2 inhibitor with Ki < 3 nM for EZH2 Y646 and EZH2 wt; 15-fold selectivity over EZH1 and >3000-fold selectivity over other HMTase.
Smiles
CCN([C@H]1CC[C@@H](CC1)N(C)CCOC)c1cc(cc(C(=O)NCc2c(C)cc(C)[nH]c2=O)c1C)C#CCN1CCOCC1
Molecular Formula
C35H51N5O4
Molecular Weight
605.81
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
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