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GSK854

Product Specifications

CAS Number

1316059-00-3

Target

Others, Apoptosis, MAPK

Related Pathways

MAPK, Apoptosis, Others

Purity

0.9891

Bioactivity

GSK854 is a highly selective and potent inhibitor of troponin I interacting kinase (TNNI3K) that inhibits myocardial infarction-injured cellular pyroptosis and apoptosis in mice, which may limit oxidative stress, injury, and adverse remodeling in the ischemic heart.

Smiles

CCS(=O)(=O)c1ccc(cc1Nc1cc(Nc2ccc(Cl)cn2)ncn1)S(=O)(=O)NC

Molecular Formula

C18H19ClN6O4S2

Molecular Weight

482.96

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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