YIL 781
Product Specifications
CAS Number
875258-85-8
Target
GHSR
Related Pathways
GPCR/G Protein
Purity
0.993
Bioactivity
YIL 781 is a selective ghrelin receptor antagonist (GHS-R1a) (Ki = 17 nM), showing a weak affinity for kinesin receptors (K = 6 μM) . YIL 781 improves glucose homeostasis in vivo and in vitro by blocking ghrelin secretion.
Smiles
O=C1C=2C(N=C(C)N1C[C@@H]3CN(C(C)C)CCC3)=CC=C(OC4=CC=C(F)C=C4)C2
Molecular Formula
C24H28FN3O2
Molecular Weight
409.5
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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