Y134
Product Specifications
CAS Number
849662-80-2
Target
Estrogen Receptor/ERR
Related Pathways
Endocrinology/Hormones
Purity
0.9998
Bioactivity
Y134 is an estrogen receptor inhibitor that is selective and orally active, exhibiting strong antagonist activity against ER? and Er? with Ki of 0.09 nM and 11.31 nM, respectively. The selectivity of Y134 for ER? is 121.1 times higher than that for ER?. Y134 inhibited the proliferation of ER positive human breast cancer cells stimulated by estrogen.
Smiles
C(=O)(C1=C(SC=2C1=CC=C(O)C2)C3=CC=C(O)C=C3)C4=CC=C(C=C4)N5CCN(C(C)C)CC5
Molecular Formula
C28H28N2O3S
Molecular Weight
472.6
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
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