MRS1220
Product Specifications
CAS Number
183721-15-5
Target
Adenosine Receptor
Related Pathways
GPCR/G Protein, Neuroscience
Purity
0.9843
Bioactivity
MRS1220, a selective and potent antagonist for the human A3 adenosine receptor (hA3AR) with a dissociation constant (Ki) of 0.59 nM, exhibits therapeutic promise for central nervous system disease research. It effectively diminishes glioblastoma tumor size and inhibits blood vessel formation in vivo.
Smiles
Clc1ccc2nc(NC(=O)Cc3ccccc3)n3nc(nc3c2c1)-c1ccco1
Molecular Formula
C21H14ClN5O2
Molecular Weight
403.82
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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