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LY 272015 hydrochloride

Product Specifications

CAS Number

172895-15-7

Target

5-HT Receptor

Related Pathways

GPCR/G Protein|||Neuroscience

Purity

0.9947

Bioactivity

LY 272015 hydrochloride is an orally active and selective 5-HT2B receptor antagonist that displays antihypertensive effects in DOCA-salt hypertensive rats.LY 272015 hydrochloride inhibits 5-HT- or BW723C86-induced ERK2 phosphorylation and attenuates MVIC and Tissue downstream cellular effects of 5HT signaling and can be used to study hepatocellular carcinoma.

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Cl.O(C1=CC=C(C=C1OC)CC2NCCC=3C=4C=C(C=CC4NC32)C)C

Molecular Formula

C21H25ClN2O2

Molecular Weight

372.89

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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