CP 154526 hydrochloride
Product Specifications
CAS Number
257639-98-8
Target
CRFR
Related Pathways
GPCR/G Protein
Purity
0.9994
Bioactivity
CP 154526 hydrochloride is a blood-brain barrier-penetrant, selective CRF1 (corticotropin-releasing factor receptor 1) antagonist (Ki = 2.7 nM) exhibiting thousands of times greater selectivity for CRF1 over CRF2, with anxiolytic and antidepressant activities.
Smiles
Cl.N=1C(=NC(=C2C1N(C=C2C)C=3C(=CC(=CC3C)C)C)N(CC)CCCC)C
Molecular Formula
C23H33ClN4
Molecular Weight
400.99
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
BNC741986-100 1x 100 µL
Tyrosinase-Related Protein-1 (TYRP-1) (Melanoma Marker) (TYRP1/1986), CF740 conjugate, 0.1mg/mL
Sign In for Pricing
View Details 
BNC941199-100 1x 100 µL
SUMO-2 (SUMO2/1199), CF594 conjugate, 0.1mg/mL
Sign In for Pricing
View Details