CP-100356 hydrochloride
Product Specifications
CAS Number
142715-48-8
Target
P-gp, BCRP
Related Pathways
Neuroscience, Membrane transporter/Ion channel
Purity
0.9919
Bioactivity
CP-100356 hydrochloride is an orally active, low micromolar dual inhibitor of MDR1 (P-gp) and BCRP, a nucleotide-derived substrate analogue that inhibits MDR1-mediated Calcein-AM and BCRP-mediated Prazosin transporters. Additionally, CP-100356 inhibits OATP1B1 and induces stomatal opening in the dark.
Smiles
Cl.COc1ccc(CCNc2nc(N3CCc4cc(OC)c(OC)cc4C3)c3cc(OC)c(OC)cc3n2)cc1OC
Molecular Formula
C31H37ClN4O6
Molecular Weight
597.1
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
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