Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

CDK8/19-IN-51

Product Specifications

CAS Number

1860885-61-5

Target

CDK

Related Pathways

Cell Cycle/Checkpoint

Purity

>99.99%

Bioactivity

CDK8/19-IN-51 is an orally active and highly effective dual inhibitor of CDK8 and CDK19, with anticancer activity. Its IC50 values for CDK8 and CDK19 are 5.1 nM and 5.6 nM, respectively. It is used in studies of colorectal and gastric cancers.

Smiles

O=C(C1=NC2=C(C=NC(N)=C2C=C1)C3=CC=C(C=C3)C=4C=NN(C4)C)N5CC(OC)C5

Molecular Formula

C23H22N6O2

Molecular Weight

414.46

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

Explore Other Products

Discover premium biology products from our extensive collection of 20M+ items

CYB5R2 Antibody, Biotin conjugated
A58050-50UG 50 µg

CYB5R2 Antibody, Biotin conjugated

Ask
View Details
1-o-Tolyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
228910-01 100 mg

1-o-Tolyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine

Ask
View Details
1-o-Tolyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
228910-02 250 mg

1-o-Tolyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine

Ask
View Details
1-o-Tolyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
228910-03 1 g

1-o-Tolyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine

Ask
View Details
1-o-Tolyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
228910-04 5 g

1-o-Tolyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine

Ask
View Details
Selenof Mouse qPCR Primer Pair (NM_053102)
MP215114 200 Reactions

Selenof Mouse qPCR Primer Pair (NM_053102)

Ask
View Details