YKL-5-124
Product Specifications
CAS Number
1957203-01-8
Target
CDK
Related Pathways
Cell Cycle/Checkpoint
Purity
0.995
Bioactivity
YKL-5-124, a potent, selective and covalent CDK7 inhibitor with an IC50 of 9.7 nM, 1300 nM and 3020 nM for CDK7/Mat1/CycH, CDK2 and CDK9 respectively, displays biochemical and cellular selectivity for CDK7 over CDK12/13.
Smiles
CN(C)C[C@@H](NC(=O)N1Cc2c(NC(=O)c3ccc(NC(=O)C=C)cc3)n[nH]c2C1(C)C)c1ccccc1
Molecular Formula
C28H33N7O3
Molecular Weight
515.61
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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