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RBN012759

Product Specifications

CAS Number

2360851-29-0

Target

PARP

Related Pathways

DNA Damage/DNA Repair|||Chromatin/Epigenetic

Purity

0.9996

Bioactivity

RBN012759 inhibits PARP14 protein with an IC50 value of 0.003 ?M and is more than 300-fold selective over all PARP family members.[2]

Smiles

O[C@H]1CC[C@@H](CC1)SCc1nc2cc(OCC3CC3)cc(F)c2c(=O)[nH]1

Molecular Formula

C19H23FN2O3S

Molecular Weight

378.46

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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