NIBR-17
Product Specifications
CAS Number
944396-88-7
Target
PI3K
Related Pathways
PI3K/Akt/mTOR signaling
Purity
0.9779
Bioactivity
NIBR-17 is a pan class I PI3K inhibitor. NIBR-17 inhibits PI3KKα, PI3KKβ, PI3KKγ, and PI3KKδ with IC50 of 1 nM, 9.2 nM, 9 nM, and 20 nM respectively.
Smiles
COc1ccc(Nc2cc(nc(n2)N2CCOCC2)-c2cnc(N)nc2)cn1
Molecular Formula
C18H20N8O2
Molecular Weight
380.4
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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