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NIBR-17

Product Specifications

CAS Number

944396-88-7

Target

PI3K

Related Pathways

PI3K/Akt/mTOR signaling

Purity

0.9779

Bioactivity

NIBR-17 is a pan class I PI3K inhibitor. NIBR-17 inhibits PI3KK?, PI3KK?, PI3KK?, and PI3KK? with IC50 of 1 nM, 9.2 nM, 9 nM, and 20 nM respectively.

Smiles

COc1ccc(Nc2cc(nc(n2)N2CCOCC2)-c2cnc(N)nc2)cn1

Molecular Formula

C18H20N8O2

Molecular Weight

380.4

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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