MDR-652
Product Specifications
CAS Number
1933528-96-1
Target
TRP/TRPV Channel
Related Pathways
Membrane transporter/Ion channel
Purity
0.9996
Bioactivity
MDR-652 is a highly specific and efficacious agonist of nonpungent transient receptor potential vanilloid 1 (TRPV1), with Ki values of 11.4 nM and 23.8 nM for hTRPV1 and rTRPV1, respectively, and EC50s of 5.05 nM and 93 nM for hTRPV1 and rTRPV1, respectively. MDR-652 is a potent topical analgesic.
Smiles
CC(C)(C)c1nc(c(CNC(=O)Nc2ccc(CO)c(F)c2)s1)-c1cccc(Cl)c1
Molecular Formula
C22H23ClFN3O2S
Molecular Weight
447.95
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
MBS6370637-01 0.1 mL
ATG7 (APG7L, Ubiquitin-like Modifier-activating Enzyme ATG7, ATG12-activating Enzyme E1 ATG7, Autophagy-related Protein 7, Ubiquitin-activating Enzyme E1-like Protein) (MaxLight 750)
Sign In for Pricing
View Details MBS6370637-02 5x 0.1 mL
ATG7 (APG7L, Ubiquitin-like Modifier-activating Enzyme ATG7, ATG12-activating Enzyme E1 ATG7, Autophagy-related Protein 7, Ubiquitin-activating Enzyme E1-like Protein) (MaxLight 750)
Sign In for Pricing
View Details 236898-01 25 mg
Cis-2-Benzyloxycarbonylaminocyclobutanecarboxylic Acid 98+%
Sign In for Pricing
View Details