What is the catalog number for MDR-652?

The catalog number for MDR-652 is T22360.

What sizes are available for MDR-652?

MDR-652 is available in the following size(s): 1 mg, 2 mg, 5 mg, 1 mL - 10 mM (in DMSO), 10 mg, 25 mg, 50 mg, 100 mg, 200 mg.

How many pack sizes does MDR-652 come in?

MDR-652 is available in 9 different pack sizes.

MDR-652 is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures MDR-652?

MDR-652 is manufactured by Molfinity.

What is the estimated delivery time for MDR-652?

Estimated delivery time for MDR-652 is approximately 10 business day(s), depending on your location.

MDR-652

Product Specifications

CAS Number

1933528-96-1

Target

TRP/TRPV Channel

Related Pathways

Membrane transporter/Ion channel

Purity

0.9996

Bioactivity

MDR-652 is a highly specific and efficacious agonist of nonpungent transient receptor potential vanilloid 1 (TRPV1), with Ki values of 11.4 nM and 23.8 nM for hTRPV1 and rTRPV1, respectively, and EC50s of 5.05 nM and 93 nM for hTRPV1 and rTRPV1, respectively. MDR-652 is a potent topical analgesic.