MDR-652
Product Specifications
CAS Number
1933528-96-1
Target
TRP/TRPV Channel
Related Pathways
Membrane transporter/Ion channel
Purity
0.9996
Bioactivity
MDR-652 is a highly specific and efficacious agonist of nonpungent transient receptor potential vanilloid 1 (TRPV1), with Ki values of 11.4 nM and 23.8 nM for hTRPV1 and rTRPV1, respectively, and EC50s of 5.05 nM and 93 nM for hTRPV1 and rTRPV1, respectively. MDR-652 is a potent topical analgesic.
Smiles
CC(C)(C)c1nc(c(CNC(=O)Nc2ccc(CO)c(F)c2)s1)-c1cccc(Cl)c1
Molecular Formula
C22H23ClFN3O2S
Molecular Weight
447.95
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
Explore Other Products
Discover premium biology products from our extensive collection of 20M+ items
P9007-53E-ML550 100 µL
PHB2 (Y128) (BAP, REA, Prohibitin-2, B Cell Receptor-associated Protein BAP37, Repressor Of Estrogen Receptor Activity, D-prohibitin) (MaxLight 550) discontinued
Ask
View Details 