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GSK3368715 3HCl

Product Specifications

CAS Number

2227587-26-8

Target

Histone Methyltransferase

Related Pathways

Chromatin/Epigenetic

Bioactivity

GSK3368715, a potent inhibitor of type I protein arginine methyltransferases (PRMT), could inhibit PRMT1, 3, 4, 6 and 8 with Kiapp vaules ranging from 1.5 to 81 nM.

Smiles

Cl.Cl.Cl.CCOCC1(COCC)CCC(CC1)c1n[nH]cc1CN(C)CCNC

Molecular Formula

C20H41Cl3N4O2

Molecular Weight

475.92

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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