CP-465022 (maleate)
Product Specifications
CAS Number
199656-46-7
Target
Others, iGluR
Related Pathways
Others, Membrane transporter/Ion channel, Neuroscience
Bioactivity
CP-465022 Maleate is a potent, selective, noncompetitive AMPA receptor antagonist with anticonvulsant activity, effectively countering the Kainate-induced response in rat cortical neurons with an IC50 of 25 nM, making it a valuable instrument for studying the involvement of AMPA receptors in various physiological and pathophysiological processes [1] [2].
Smiles
OC(=O)\C=C/C(O)=O.CCN(CC)Cc1cccc(\C=C\c2nc3ccc(F)cc3c(=O)n2-c2ccccc2Cl)n1
Molecular Formula
C30H28ClFN4O5
Molecular Weight
579.02
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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