Drinabant
Product Specifications
CAS Number
358970-97-5
Target
Cannabinoid Receptor
Related Pathways
GPCR/G Protein
Purity
0.9992
Bioactivity
Drinabant (AVE-1625) is an orally active CB1 receptor antagonist. Drinabant inhibits the agonist-stimulated calcium signal with IC50 values of 25 nM and 10 nM for the hCB1-R and rCB1-R, respectively, and is ineffective for the hCB2-R.
Smiles
C(N1CC(N(S(C)(=O)=O)C2=CC(F)=CC(F)=C2)C1)(C3=CC=C(Cl)C=C3)C4=CC=C(Cl)C=C4
Molecular Formula
C23H20Cl2F2N2O2S
Molecular Weight
497.38
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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