A 784168
Product Specifications
CAS Number
824982-41-4
Target
TRP/TRPV Channel, Others
Related Pathways
Membrane transporter/Ion channel, Others
Bioactivity
A-784168, a potent and orally active inhibitor of vanilloid receptor type 1 (TRPV1), acts on a ligand-gated nonselective cation channel pivotal in integrating pain stimuli including endogenous lipids, capsaicin, heat, and low pH. It demonstrates commendable central nervous system (CNS) penetration upon oral administration [1].
Smiles
C(F)(F)(F)C1=C(N=CC=C1)N2CCC(C(NC3=CC=C(S(C(F)(F)F)(=O)=O)C=C3)=O)=CC2
Molecular Formula
C19H15F6N3O3S
Molecular Weight
479.4
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
More Discoveries
Explore Other Products
Browse additional items from our catalog
K0038108 1.0 µg DNA
ACTN4 sgRNA CRISPR/Cas9 All-in-One Lentivector (Human) (Target 3)
Sign In for Pricing
View Details 
465685-01 1 mg
S-N- (4- ((3-Cyano-1- ((3,5-dimethylisoxazol-4-yl) methyl) -1H-indol-5-yl) oxy) phenyl) pyrrolidine-2-carboxamide
Sign In for Pricing
View Details 465685-02 2.5 mg
S-N- (4- ((3-Cyano-1- ((3,5-dimethylisoxazol-4-yl) methyl) -1H-indol-5-yl) oxy) phenyl) pyrrolidine-2-carboxamide
Sign In for Pricing
View Details 
