PF-4981517
Product Specifications
CAS Number
1390637-82-7
Target
Cytochromes P450
Related Pathways
Metabolism
Purity
0.9983
Bioactivity
PF-4981517 (CYP3cide) is a efficient, specific and time-dependent inhibitor of cytochrome P4503A4 (CYP3A4) . The IC 50 values for CYP3A activity are 0.03 μM,17 μM, and 71 μM for CYP3A4, CYP3A5, and CYP3A7, respectively. PF-4981517 is able to be used to distinguish the contributions of CYP3A4 versus CYP3A5 on drug Metabolism.
Smiles
Cc1ccc(cc1)-c1c(cnn1C)-c1nn(C)c2ncnc(N3CC[C@@H](C3)N3CCCCC3)c12
Molecular Formula
C26H32N8
Molecular Weight
456.59
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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