PF-4981517
Product Specifications
CAS Number
1390637-82-7
Target
Cytochromes P450
Related Pathways
Metabolism
Purity
0.9983
Bioactivity
PF-4981517 (CYP3cide) is a efficient, specific and time-dependent inhibitor of cytochrome P4503A4 (CYP3A4) . The IC 50 values for CYP3A activity are 0.03 ?M,17 ?M, and 71 ?M for CYP3A4, CYP3A5, and CYP3A7, respectively. PF-4981517 is able to be used to distinguish the contributions of CYP3A4 versus CYP3A5 on drug Metabolism.
Smiles
Cc1ccc(cc1)-c1c(cnn1C)-c1nn(C)c2ncnc(N3CC[C@@H](C3)N3CCCCC3)c12
Molecular Formula
C26H32N8
Molecular Weight
456.59
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Product Datasheet
https://www.targetmol.com/attachment/DataSheet/B17513AE-31ED-41E1-BB0D-A4D0C5593176/T21548
Available Sizes
Curated Selection
Explore Other Products
Discover premium biology products from our extensive collection of 20M+ items
![Rabbit Polyclonal NANOS1 Antibody [DyLight 594]](https://cdn.genprice.uk/genprice/genprice5.png)
