GYKI-52466
Product Specifications
CAS Number
102771-26-6
Target
Others|||iGluR
Related Pathways
Others|||Neuroscience|||Membrane transporter/Ion channel
Bioactivity
GYKI-52466 is a selective non-competitive AMPA receptor antagonist (IC50 values are 10-20, ~ 450 and >50 ?M for AMPA-, kainate- and NMDA-induced responses, respectively) used as a Skeletal muscle relaxant, orally active anticonvulsant, neuroprotective and anxiolytic in vivo.
Smiles
CC=1CC2=C(C(=NN1)C3=CC=C(N)C=C3)C=C4C(=C2)OCO4
Molecular Formula
C17H15N3O2
Molecular Weight
293.32
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
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