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ETP-46464

Product Specifications

CAS Number

1345675-02-6

Target

DNA-PK, ATM/ATR, mTOR, PI3K

Related Pathways

PI3K/Akt/mTOR signaling, DNA Damage/DNA Repair

Purity

0.9956

Bioactivity

ETP-46464 is an effective and specific ATR inhibitor (IC50: 25 nM) .

Smiles

CC(C)(C#N)c1ccc(cc1)N1C(=O)OCc2cnc3ccc(cc3c12)-c1cnc2ccccc2c1

Molecular Formula

C30H22N4O2

Molecular Weight

470.52

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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