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APY0201

Product Specifications

CAS Number

1232221-74-7

Target

PI3K, Interleukin

Related Pathways

PI3K/Akt/mTOR signaling, Immunology/Inflammation

Purity

0.9974

Bioactivity

APY0201 is a effective, highly specific, ATP-competitive PIKfyve inhibitor (IC50: 5.2 nM) . It can interrupt the conversion of phosphatidylinositol 3-phosphate (PtdIns3P) to PtdIns (3, 5) P2.

Smiles

Cc1cccc(\C=N\Nc2cc(N3CCOCC3)n3nc(cc3n2)-c2ccncc2)c1

Molecular Formula

C23H23N7O

Molecular Weight

413.48

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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