APY0201
Product Specifications
CAS Number
1232221-74-7
Target
PI3K, Interleukin
Related Pathways
PI3K/Akt/mTOR signaling, Immunology/Inflammation
Purity
0.9974
Bioactivity
APY0201 is a effective, highly specific, ATP-competitive PIKfyve inhibitor (IC50: 5.2 nM) . It can interrupt the conversion of phosphatidylinositol 3-phosphate (PtdIns3P) to PtdIns (3, 5) P2.
Smiles
Cc1cccc(\C=N\Nc2cc(N3CCOCC3)n3nc(cc3n2)-c2ccncc2)c1
Molecular Formula
C23H23N7O
Molecular Weight
413.48
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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