CL 316243
CL316243 is a highly potent selective β3-adrenoceptor agonist with a EC50 of 3 nM, but is an extremely poor to β1/2- receptors[1].CL316243 is a effective stimulant of adipocyte lipolysis and increases brown adipose tissue thermogenesis and metabolic rate[2]. CL316243 has the potential for the treatment obesity, diabetes and urge urinary incontinence[3].
Product Specifications
CAS Number
138908-40-4
Product Name Alternative
Saponin
UNSPSC
12352005
Target
Adrenergic Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Metabolic Disease
Assay Protocol
https://www.medchemexpress.com/cl-316243.html
Purity
99.98
Solubility
DMSO : 17.5 mg/mL (ultrasonic; warming; heat to 60°C) |H2O : 4.55 mg/mL (ultrasonic; warming; adjust pH to 12 with 1 M NaOH; heat to 60°C)
Smiles
O=C(C1(C(O[Na])=O)OC2=CC=C(C[C@H](NC[C@@H](C3=CC=CC(Cl)=C3)O)C)C=C2O1)O[Na]
Molecular Formula
C20H18ClNNa2O7
Molecular Weight
465.79
References & Citations
Shipping Conditions
Room Temperature
Storage Conditions
4°C (Powder, sealed storage, away from moisture)
Scientific Category
Reference compound1
Clinical Information
Phase 2
Isoform
β adrenergic receptor
Available Sizes
Frequently Asked Questions
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