GSK-5959

Product Specifications

CAS Number

901245-65-6

Target

Epigenetic Reader Domain

Related Pathways

Chromatin/Epigenetic

Purity

0.9877

Bioactivity

GSK-5959 is an effective, specific and cell permeable BRPF1 bromodomain inhibitor (IC50: ~80 nM) . The selectivity of GSK-5959 for BRPF1 is >100-fold over a panel of 35 other bromodomains, including BRPF2/3 and BET family bromodomains.

Smiles

COc1ccccc1C(=O)Nc1cc2n(C)c(=O)n(C)c2cc1N1CCCCC1

Molecular Formula

C22H26N4O3

Molecular Weight

394.47

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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