AM251
Product Specifications
CAS Number
183232-66-8
Target
GPCR, Cannabinoid Receptor
Related Pathways
GPCR/G Protein, Endocrinology/Hormones
Purity
0.9879
Bioactivity
AM251 is a effective CB1 receptor antagonist (IC50/Ki: 8 /7.49 nM) that displays 306-fold selectivity over CB2 receptors; also effective GPR55 agonist (EC50: 39 nM) .
Smiles
CC1=C(N(N=C1C(NN2CCCCC2)=O)C3=C(Cl)C=C(Cl)C=C3)C4=CC=C(I)C=C4
Molecular Formula
C22H21Cl2IN4O
Molecular Weight
555.24
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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