BX-912
Product Specifications
CAS Number
702674-56-4
Target
PKA, PDK, Chk, VEGFR, Apoptosis, CDK
Related Pathways
Angiogenesis, Apoptosis, PI3K/Akt/mTOR signaling, Tyrosine Kinase/Adaptors, Cell Cycle/Checkpoint
Purity
0.9934
Bioactivity
BX-912 is a specific inhibitor of 3-Phosphoinositide-dependent Kinase-1 (PDK1, IC50: 12 nM) . The selectivity of BX-912 is more 10 fold than C-Kit, EGFR, PKA, PKC etc.
Smiles
Brc1cnc(Nc2cccc(NC(=O)N3CCCC3)c2)nc1NCCc1cnc[nH]1
Molecular Formula
C20H23BrN8O
Molecular Weight
471.35
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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