BRD7-IN-1
Product Specifications
CAS Number
2448414-48-8
Target
Epigenetic Reader Domain
Related Pathways
Chromatin/Epigenetic
Purity
0.9895
Bioactivity
BRD7-IN-1, a modified derivative of BI7273 (BRD7/9 inhibitor), forms PROTAC VZ185 via linkage to a VHL ligand, demonstrating potent activity against BRD7/9 with DC50 values of 4.5 and 1.8 nM, respectively [1].
Smiles
Cl.Cl.COc1cc(cc(OC)c1CN1CCNCC1)-c1cn(C)c(=O)c2cnccc12
Molecular Formula
C22H28Cl2N4O3
Molecular Weight
467.39
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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