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PD153035 hydrochloride

Product Specifications

CAS Number

183322-45-4

Target

EGFR

Related Pathways

Angiogenesis, JAK/STAT signaling, Tyrosine Kinase/Adaptors

Purity

>99.99%

Bioactivity

PD153035 hydrochloride (ZM 252868) is a effective and selective inhibitor of EGFR (Ki: 5.2 pM, IC50: 29 pM) ; few influence against FGFR, PGDFR, InsR, CSF-1, and Src.

Smiles

Cl.COc1cc2ncnc(Nc3cccc(Br)c3)c2cc1OC

Molecular Formula

C16H15BrClN3O2

Molecular Weight

396.67

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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