YM022
Product Specifications
CAS Number
145084-28-2
Target
CCR
Related Pathways
GPCR/G Protein|||Immunology/Inflammation|||Microbiology/Virology
Bioactivity
YM022 is a highly effective and selective gastrin/cholecystokinin (CCK) -B receptor antagonist. YM022 can inhibit gastrin-induced gastric acid secretion and histidine decarboxylase activation in vivo. YM022 shows the Ki values of 68 pM and 63 nM for CCK-B and CCK-A receptor, respectively.
Smiles
Cc1cccc(NC(=O)N[C@@H]2N=C(c3ccccc3)c3ccccc3N(CC(=O)c3ccccc3C)C2=O)c1
Molecular Formula
C32H28N4O3
Molecular Weight
516.59
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
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