VU0529331
Product Specifications
CAS Number
1286725-49-2
Target
Others, Potassium Channel
Related Pathways
Others, Membrane transporter/Ion channel
Bioactivity
VU0529331 is a modestly selective non-GIRK1-containing G protein-gated, inwardly-rectifying, potassium channel activator (EC50s: 5.1 μM and 5.2 μM for GIRK2 and GIRK1/2 in HEK293 cells, respectively), and is also effective on the GIRK4 homomeric channel.
Smiles
Cc1ccc(cc1C)-n1nc2CN(Cc2c1-n1cccc1)C(=O)c1cnccn1
Molecular Formula
C22H20N6O
Molecular Weight
384.43
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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