What is the catalog number for VU0463271?

The catalog number for VU0463271 is T17243.

What sizes are available for VU0463271?

VU0463271 is available in the following size(s): 5 mg, 1 mL - 10 mM (in DMSO), 10 mg, 25 mg, 50 mg, 100 mg, 200 mg.

How many pack sizes does VU0463271 come in?

VU0463271 is available in 7 different pack sizes.

Is VU0463271 in stock?

VU0463271 is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures VU0463271?

VU0463271 is manufactured by Molfinity.

What is the estimated delivery time for VU0463271?

Estimated delivery time for VU0463271 is approximately 10 business day(s), depending on your location.

VU0463271

Product Specifications

CAS Number

1391737-01-1

Target

Potassium Channel

Related Pathways

Membrane transporter/Ion channel

Purity

0.9975

Bioactivity

VU0463271 (N-Cyclopropyl-N- (4-methyl-2-thiazolyl) -2-[ (6-phenyl-3-pyridazinyl) thio]acetamide) is a potent and selective antagonist of the neuronal-specific potassium-chloride cotransporter 2 (KCC2), with an IC50 of 61 nM and >100-fold selectivity versus the closely related Na-K-2Cl cotransporter 1 (NKCC1) and no activity in a larger panel of GPCRs, ion channels, and transporters.