UPGL00004
Product Specifications
CAS Number
1890169-95-5
Target
Glutaminase
Related Pathways
Proteases/Proteasome
Purity
0.9793
Bioactivity
UPGL00004 is a potent glutaminase C (GAC) inhibitor with an IC50 of 29 nM. Kd of UPGL00004 for GAC was 27 nM. UPGL00004 has a strong inhibitory effect on the proliferation of highly aggressive triple negative breast cancer cell lines.
Smiles
O=C(Cc1ccccc1)Nc1nnc(NC2CCN(CC2)c2nnc(NC(=O)Cc3ccccc3)s2)s1
Molecular Formula
C25H26N8O2S2
Molecular Weight
534.66
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
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