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Tilfrinib

Product Specifications

CAS Number

1600515-49-8

Target

BTK

Related Pathways

Angiogenesis, Tyrosine Kinase/Adaptors

Purity

0.9973

Bioactivity

Tilfrinib is an effective and selective inhibitor of breast tumor kinase (Brk, IC50 = 3.15 nM) which displays anti-proliferative and anti-tumor activities.

Smiles

Oc1cccc(Nc2ccnc3[nH]c4ccccc4c23)c1

Molecular Formula

C17H13N3O

Molecular Weight

275.3

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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